Ara mostrant els elements 1-10 de 21
Garcia Subirats, Maria (Data de defensa: 2015-12-16)
El problema de la resistència bacteriana ha esdevingut un problema de salut pública global. Cada cop apareixen més soques bacterianes resistents a dos o més fàrmacs i és especialment preocupant la manca ...
Granados Ramírez, Carmen Giovana (Data de defensa: 2008-01-16)
1) "Diseño, síntesis y caracterización de inhibidores de la fusión de VIH-1 análogos del péptido C34 de gp41 con D aminoácido"<br/><br/>En el proceso de fusión del virus del VIH-1 a la célula diana ...
Garcia Pindado, Júlia (Data de defensa: 2017-05-12)
The present thesis is based on the development and optimization of a solid-phase strategy to prepare biaryl bicyclic pentapeptides. Suzuki-Miyaura cross-coupling reactions were used to obtain the biaryl ...
Matas Moya, Sonia (Data de defensa: 2013-12-02)
En la present tesi doctoral s’ha plantejat com un dels principals objectius desenvolupar un sistema de diagnòstic in vitro per a detectar al∙lèrgies a fàrmacs β‐lactàmics, i més concretament contra ...
Messeguer Escriche, Joaquim (Data de defensa: 2007-07-17)
La recerca en el camp del desenvolupament de fàrmacs peptídics i peptidomimètics ha experimentat una evolució important durant els darrers anys. Els fàrmacs peptídics sovint presenten baixa disponibilitat ...
Isidro Llobet, Albert (Data de defensa: 2008-05-13)
The increasing importance of peptides as drugs creates the necessity of new methodologies for the synthesis of complex peptides. This PhD thesis has been focused on the development of new protecting ...
Tapia Pérez, Lucía (Data de defensa: 2021-10-01)
This PhD thesis lays on the field of supramolecular chemistry. In this field, there is a huge interest in the development of cage-like compounds able to bind biologically relevant molecules inside their ...
Martín-Gago, Pablo (Data de defensa: 2013-10-11)
Somatostatin, a peptidic hormone also known as somatotropin release-inhibiting factor (SRIF), is implicated in multiple biological functions, mediated by direct interaction of the peptide with a family ...
Díaz Perlas, Cristina (Data de defensa: 2018-03-07)
Peptides play a critical role in human physiology and harbour a huge potential as therapeutic agents. In this thesis, new peptides have been discovered as ligands for the epidermal growth factor (EGF) ...
Fernández-Llamazares Onrubia, Ana Iris (Data de defensa: 2013-12-09)
Backbone N-methylation is becoming an increasingly important tool in peptide drug design, and has been widely used to optimize the activity and selectivity of peptide ligands as a result of conformational ...